BDBM320489 US10174035, Compound 35::[2-(1-Methyl-1H-pyrazol-4-yl)-6-(morpholin-4-yl)-9H-purin-8-yl](4-phenylpiperidin-1-yl)methanone

SMILES Cn1cc(cn1)-c1nc(N2CCOCC2)c2nc([nH]c2n1)C(=O)N1CCC(CC1)c1ccccc1

InChI Key InChIKey=PWCLCQRTWAKAFQ-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 320489   

TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Daiichi Sankyo

US Patent

LigandBDBM320489([2-(1-Methyl-1H-pyrazol-4-yl)-6-(morpholin-4-yl)-9...)Copy SMILESCopy InChI

Affinity DataIC50: 17nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
5/16/2019
Entry Details
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