BDBM320580 US10174035, Compound 123::{6-Fluoro-7-(morpholin-4-yl)-5-[3-(trifluoromethyl)-1H-pyrazol-4-yl]-3H-imidazo[4,5-b]pyridin-2-yl}[4-(morpholin-4-yl)piperidin-1-yl]methanone

SMILES Fc1c(nc2[nH]c(nc2c1N1CCOCC1)C(=O)N1CCC(CC1)N1CCOCC1)-c1c[nH]nc1C(F)(F)F

InChI Key InChIKey=CWRCVMJHKVLTQZ-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 320580   

TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Daiichi Sankyo

US Patent

LigandBDBM320580(US10174035, Compound 123 | {6-Fluoro-7-(morpholin-...)Copy SMILESCopy InChI

Affinity DataIC50: 4nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
5/16/2019
Entry Details
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