BDBM320586 1-Methyl-4-(1-{[5-(1-methyl-1H-pyrazol-4-yl)-7-(morpholin-4-yl)-3H-imidazo[4,5-b]pyridin-2-yl]carbonyl}azetidin-3-yl)piperazin-2-one::US10174035, Compound 129

SMILES CN1CCN(CC1=O)C1CN(C1)C(=O)c1nc2c(cc(nc2[nH]1)-c1cnn(C)c1)N1CCOCC1

InChI Key InChIKey=XHQJLOKZQICOMG-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 320586   

TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Daiichi Sankyo

US Patent

LigandBDBM320586(US10174035, Compound 129 | 1-Methyl-4-(1-{[5-(1-me...)Copy SMILESCopy InChI

Affinity DataIC50: 10nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
5/16/2019
Entry Details
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