BDBM3253 (1R,2R)-2-[(4-hydroxybenzene)amido]cyclopentyl 4-{[2-(ethoxycarbonyl)-6-hydroxyphenyl]carbonyl}-3,5-dihydroxybenzoate::Balanol Benzophenone Ester Analog 15

SMILES CCOC(=O)c1cccc(O)c1C(=O)c1c(O)cc(cc1O)C(=O)O[C@@H]1CCC[C@H]1NC(=O)c1ccc(O)cc1

InChI Key InChIKey=MGLBGUZLARZAOR-UHFFFAOYSA-N

Data  5 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 3253   

TargetProtein kinase C alpha type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3253((1R,2R)-2-[(4-hydroxybenzene)amido]cyclopentyl 4-{...)
Affinity DataIC50: 920nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C beta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3253((1R,2R)-2-[(4-hydroxybenzene)amido]cyclopentyl 4-{...)
Affinity DataIC50: 1.60E+3nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C delta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3253((1R,2R)-2-[(4-hydroxybenzene)amido]cyclopentyl 4-{...)
Affinity DataIC50: 67nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C epsilon type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3253((1R,2R)-2-[(4-hydroxybenzene)amido]cyclopentyl 4-{...)
Affinity DataIC50: 660nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C eta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM3253((1R,2R)-2-[(4-hydroxybenzene)amido]cyclopentyl 4-{...)
Affinity DataIC50: 52nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article