BDBM331642 Preparation of 2-(4-(1H-pyrrolo[2,3-b]pyridin-5-yl)phenyl)-N-(5-(1-(trifluoromethyl)cyclopropyl)isoxazol-3-yl)acetamide::US9725465, Example 18

SMILES FC(F)(F)C1(CC1)c1cc(NC(=O)Cc2ccc(cc2)-c2cnc3[nH]ccc3c2)no1

InChI Key InChIKey=KGIGUJRAZWOBAK-UHFFFAOYSA-N

Data  1 Kd

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 331642   

TargetMast/stem cell growth factor receptor Kit(Human)
Ambit Biosciences

US Patent
LigandPNGBDBM331642(US9725465, Example 18 | Preparation of 2-(4-(1H-py...)
Affinity DataKd: <5nMAssay Description:Competition binding assays used herein were developed, validated and performed as described in Fabian et al., Nature Biotechnology 2005, 23, 329-336....More data for this Ligand-Target Pair
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Date in BDB:
6/12/2019
Entry Details
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