BDBM345782 5-[2-Methoxy-6-(1-phenyl- ethylamino)-pyrimidin-4-yl]-1- methyl-1H-pyridin-2-one::US10202360, Example 327

SMILES COc1nc(NC(C)c2ccccc2)cc(n1)-c1ccc(=O)n(C)c1

InChI Key InChIKey=KPNBDLOIFKPLSF-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 345782   

TargetCREB-binding protein(Human)
Celgene Quanticel Research

US Patent
LigandPNGBDBM345782(US10202360, Example 327 | 5-[2-Methoxy-6-(1-phenyl...)
Affinity DataIC50: 500nMAssay Description:Determination of the IC50 for the CREBBP inhibitors disclosed herein was performed as follows: CREBBP was cloned and expressed in E. Coli as His-tag ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent