BDBM355735 Azetidin-1-yl[3-(4-chloro-2,5-difluorophenyl)-3H-imidazo[4,5-b]pyridin-2-yl]methanone, trifluoroacetate salt::US9815832, 12

SMILES Fc1cc(c(F)cc1Cl)-n1c(nc2cccnc12)C(=O)N1CCC1

InChI Key InChIKey=XSRUKFNHJGPNOA-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 355735   

LigandPNGBDBM355735(US9815832, 12 | Azetidin-1-yl[3-(4-chloro-2,5-difl...)
Affinity DataIC50: 99.4nMAssay Description:The PDE4B and 4D assays use scintillation proximity assay (SPA) technology to measure the inhibition of human recombinant PDE4B and PDE4D enzyme acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2019
Entry Details
US Patent

LigandPNGBDBM355735(US9815832, 12 | Azetidin-1-yl[3-(4-chloro-2,5-difl...)
Affinity DataIC50: 1.52E+3nMAssay Description:The PDE4B and 4D assays use scintillation proximity assay (SPA) technology to measure the inhibition of human recombinant PDE4B and PDE4D enzyme acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2019
Entry Details
US Patent