BDBM357907 (E)-2-Amino-8-(2-cyclopentylvinyl)-5-oxo-5H-chromeno[2,3-b]pyridine-3-carboxylic acid::US10214536, Compound 253b

SMILES Nc1nc2oc3cc(\C=C\C4CCCC4)ccc3c(=O)c2cc1C(O)=O

InChI Key InChIKey=RPCFCHGKANWILU-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 357907   

TargetSerine/threonine-protein kinase TBK1(Human)
University of Michigan

US Patent
LigandPNGBDBM357907(US10214536, Compound 253b | (E)-2-Amino-8-(2-cyclo...)
Affinity DataIC50: 1.49E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent