BDBM368508 1-ethyl-4-fluoro-N-(1H- pyrazolo[4,3-b]pyridin-3 yl)isoquinolin-6-amine::US10227343, Example 41

SMILES CCc1ncc(F)c2cc(Nc3n[nH]c4cccnc34)ccc12

InChI Key InChIKey=IRPOGRSJDARHBD-UHFFFAOYSA-N

Data  1 EC50

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 368508   

TargetMetabotropic glutamate receptor 4(Human)
Vanderbilt University

US Patent
LigandPNGBDBM368508(1-ethyl-4-fluoro-N-(1H- pyrazolo[4,3-b]pyridin-3 y...)
Affinity DataEC50:  22nMAssay Description:The disclosed compounds and compositions can be evaluated for their ability to act as a potentiator of metabotropic glutamate receptor activity, in p...More data for this Ligand-Target Pair
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Date in BDB:
12/27/2019
Entry Details
US Patent