BDBM369009 N-[4-(6,7-dimethoxyquinazolin-4-yl)-2- fluoro-phenyl]-4-methoxy- benzenesulfonamide::US10227357, Compound P-0273

SMILES COc1ccc(cc1)S(=O)(=O)Nc1ccc(cc1F)-c1ncnc2cc(OC)c(OC)cc12

InChI Key InChIKey=JDMJXCTWASLKHU-UHFFFAOYSA-N

Data  1 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 369009   

LigandPNGBDBM369009(US10227357, Compound P-0273 | N-[4-(6,7-dimethoxyq...)
Affinity DataKi:  500nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2019
Entry Details
US Patent