BDBM3785 N-(3-bromophenyl)-3,7-dithia-5,10,12-triazatricyclo[6.4.0.0^{2,6}]dodeca-1(8),2(6),4,9,11-pentaen-9-amine::Thiazolothieno[3,2-d]pyrimidine deriv. 76

SMILES Brc1cccc(Nc2ncnc3c2sc2ncsc32)c1

InChI Key InChIKey=RLAGSKIPOCVMQK-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 3785   

TargetEpidermal growth factor receptor(Human)
Parke-Davis Pharmaceutical Research

LigandPNGBDBM3785(N-(3-bromophenyl)-3,7-dithia-5,10,12-triazatricycl...)
Affinity DataIC50: 40nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2005
Entry Details Article
PubMed