BDBM393275 5-(4- fluorobenzenesulfon- amidomethyl)-6- methyl-N-[(2-methyl- 1,3-thiazol-5- yl)methyl]pyrazine-2- carboxamide::US9963434, Table 12.218

SMILES Cc1ncc(CNC(=O)c2cnc(CNS(=O)(=O)c3ccc(F)cc3)c(C)n2)s1

InChI Key InChIKey=DABGPNSCWLSWOH-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 393275   

TargetGlutamate receptor ionotropic, NMDA 2A(Human)
Luc Therapeutics

US Patent
LigandPNGBDBM393275(US9963434, Table 12.218 | 5-(4- fluorobenzenesulfo...)
Affinity DataIC50: 137nMAssay Description:Cell Culture and plating: HEK293 cells expressing NR1/NR2A (Chantest, Cleveland, Ohio) were grown to 70-80% confluency as an adherent monolayer in st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2020
Entry Details
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