BDBM410094 N-(Cyclopropylsulfonyl)-2-((3R,4S or 3S,4R)-4-hydroxy-3-((5-(2-methylthiazol-5-yl)pyridin-2-yl)methyl)chroman-7-yl)benzamide::US10370368, Example 11

SMILES Cc1ncc(s1)-c1ccc(C[C@@H]2COc3cc(ccc3[C@H]2O)-c2ccccc2C(=O)NS(=O)(=O)C2CC2)nc1

InChI Key InChIKey=ULEIBGDPYYYCTK-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 410094   

TargetLeukotriene B4 receptor 1(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM410094(N-(Cyclopropylsulfonyl)-2-((3R,4S or 3S,4R)-4-hydr...)
Affinity DataEC50:  391nMAssay Description:The ability of compounds to antagonize the human BLT1 receptor was determined using a kit to measure changes in intracellular cyclic AMP levels (cAMP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
US Patent