BDBM447126 1-[3-[6-[3- (hydroxymethyl) phenyl]imidazo [1,2-b]pyridazin- 3-yl]phenyl] ethanone::US10688093, Compound 828_4145_0291::US10688093, Compound BF000726471 (828_4145_0291)::US11701353, Compound 828_4145_0291

SMILES CC(=O)c1cccc(c1)-c1cnc2ccc(nn12)-c1cccc(CO)c1

InChI Key InChIKey=AQQNAHOSRQOSPU-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 447126   

TargetTyrosine-protein kinase Fyn(Human)
Pathways Neuro Pharma

US Patent
LigandPNGBDBM447126(US10688093, Compound BF000726471 (828_4145_0291) |...)
Affinity DataIC50: 179nMAssay Description:The assay procedure determines the IC50 of each potential FYN kinase inhibitor by measuring the enzyme catalyzed ATP-dependent phosphorylation of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details
US Patent

TargetTyrosine-protein kinase Fyn(Human)
Pathways Neuro Pharma

US Patent
LigandPNGBDBM447126(US10688093, Compound BF000726471 (828_4145_0291) |...)
Affinity DataIC50: 291nMAssay Description:The assay procedure determines the IC50 of each potential FYN kinase inhibitor by measuring the enzyme catalyzed ATP-dependent phosphorylation of the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details
US Patent