BDBM455984 4-(3- (cyclopropylethynyl)-2- (1-(hydroxyamino)-1- oxo-3-phenylpropan-2- yl)-2H-pyrazolo[3,4- c]pyridin-7-yl)-N- methylbenzamide::US10723705, No. I-0141

SMILES CNC(=O)c1ccc(cc1)-c1nccc2c(C#CC3CC3)n(nc12)C(Cc1ccccc1)C(=O)NO

InChI Key InChIKey=PDBYKEPMYVCTBZ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 455984   

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandPNGBDBM455984(4-(3- (cyclopropylethynyl)-2- (1-(hydroxyamino)-1-...)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
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