BDBM481637 N1,N4-dibenzyl-N1-ethyl-N4-(2- fluorobenzyl)benzene-1,4- disulfonamide::US10913710, Compound 49

SMILES CCN(Cc1ccccc1)S(=O)(=O)c1ccc(cc1)S(=O)(=O)N(Cc1ccccc1)Cc1ccccc1F

InChI Key InChIKey=RNXUVUTXBUZTEX-UHFFFAOYSA-N

Data  1 Kd

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 481637   

TargetRetinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit delta(Human)
Max-Planck-Gesellschaft Zur Forderung Der Wissenschaften

US Patent
LigandPNGBDBM481637(N1,N4-dibenzyl-N1-ethyl-N4-(2- fluorobenzyl)benzen...)
Affinity DataKd:  16nMAssay Description:Binding to PDEδ was validated and quantified by means of a displacement assay employing a fluorescent-tagged analog of the HMG-CoA reductase inh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2021
Entry Details
US Patent