BDBM483920 US10927106, Compound PST-129::US10927106, Compound PST-131

SMILES COc1ccc(Oc2ccncc2-c2nc3cc(OC)ccc3s2)c(Cl)c1

InChI Key InChIKey=ZUYVNNKQOWXSSK-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 483920   

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Pharmasum Therapeutics

US Patent
LigandPNGBDBM483920(US10927106, Compound PST-129 | US10927106, Compoun...)
Affinity DataIC50: 351nMAssay Description:The principal method utilized is a radioactive filter binding assay using 33P ATP This method is sensitive, accurate and provides a direct measure of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Pharmasum Therapeutics

US Patent
LigandPNGBDBM483920(US10927106, Compound PST-129 | US10927106, Compoun...)
Affinity DataIC50: 3.86E+3nMAssay Description:The principal method utilized is a radioactive filter binding assay using 33P ATP This method is sensitive, accurate and provides a direct measure of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent