BDBM492903 US10981899, Example RU-0207148

SMILES Oc1ccc(Br)cc1C(=O)C1=CC(C(=O)C(=C1)C#N)c1ccccc1Cl

InChI Key InChIKey=QKZGTUNWBCNABC-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 492903   

TargetAdenylate cyclase type 10(Human)
Cornell University

US Patent
LigandPNGBDBM492903(US10981899, Example RU-0207148)
Affinity DataIC50: 4.40E+3nMAssay Description:INS-1E insulinoma cells were incubated in 2.5 mM glucose Krebs-Ringer buffer (pH 7.5) supplemented with 2 mM sodium bicarbonate, 10 mM HEPES, and 0.1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2021
Entry Details
US Patent

TargetAdenylate cyclase type 10(Human)
Cornell University

US Patent
LigandPNGBDBM492903(US10981899, Example RU-0207148)
Affinity DataIC50: 5.70E+3nMAssay Description:The RapidFire 365 High-throughput MS System (Agilent Technologies; RF-MSS) can process samples every 15 seconds allowing analysis of a 384 well plate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2021
Entry Details
US Patent