BDBM499604 US11020395, Example 200.0::US11020395, Example 201.0

SMILES CO[C@@H]([C@H](C)S(=O)(=O)Nc1nnc(C2CC3(CC3)C2)n1-c1c(OC)ncnc1OC)c1ncc(C)cn1

InChI Key InChIKey=XZHNJVYHSDWVND-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 499604   

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM499604(US11020395, Example 201.0 | US11020395, Example 20...)
Affinity DataEC50:  4.60nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV -3 expression vector (Si...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2021
Entry Details
US Patent

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM499604(US11020395, Example 201.0 | US11020395, Example 20...)
Affinity DataEC50:  11nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV -3 expression vector (Si...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2021
Entry Details
US Patent