BDBM50007966 CHEMBL420022::Tyr-Gly(psi)CH2O-Gly-PheLeu-NH2

SMILES CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)COCCNC(=O)[C@@H](N)Cc1ccc(O)cc1)C(N)=O

InChI Key InChIKey=UXGIOYDDYMEKLJ-UHFFFAOYSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50007966   

TargetMu-type opioid receptor(Rat)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50007966(CHEMBL420022 | Tyr-Gly(psi)CH2O-Gly-PheLeu-NH2)
Affinity DataKi:  1.38E+3nMAssay Description:Binding affinity to opioid receptor mu was determined in rat brain using [3H]DAGO as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50007966(CHEMBL420022 | Tyr-Gly(psi)CH2O-Gly-PheLeu-NH2)
Affinity DataKi:  9.20E+3nMAssay Description:Binding affinity to opioid receptor delta was determined in rat brain using [3H]DSTBULET as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed