BDBM50011182 CHEMBL3260318

SMILES Cc1cc(C)nc(Nc2cc(N[C@@H]3CCCC[C@@H]3N)ccc2C(N)=O)c1

InChI Key InChIKey=FHLLUBJCTSMNCQ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50011182   

TargetTyrosine-protein kinase SYK(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50011182(CHEMBL3260318)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of human recombinant SYK by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50011182(CHEMBL3260318)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of full-length GST-tagged human Syk preincubated for 10 mins followed by peptide substrate/ATP addition measured after 45 mins by TR-FRET ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2016
Entry Details Article
PubMed