BDBM50017517 1-(8-Chloro-5-ethylidene-5H-dibenzo[a,d]cyclohepten-10-yl)-4-methyl-piperazine::CHEMBL308843

SMILES C\C=C1\c2ccccc2C=C(N2CCN(C)CC2)c2cc(Cl)ccc12

InChI Key InChIKey=GPGQEGGSDSKZFR-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50017517   

TargetD(1A) dopamine receptor(Rat)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50017517(CHEMBL308843 | 1-(8-Chloro-5-ethylidene-5H-dibenzo...)
Affinity DataIC50: 305nMAssay Description:Binding activity against Dopamine receptor D1 in rat brain, using [3H]SCH-23390 as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50017517(CHEMBL308843 | 1-(8-Chloro-5-ethylidene-5H-dibenzo...)
Affinity DataIC50: 2.60E+3nMAssay Description:Binding activity against muscarinic acetylcholine receptor in rat brain using [3H]QNB as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50017517(CHEMBL308843 | 1-(8-Chloro-5-ethylidene-5H-dibenzo...)
Affinity DataIC50: 6.97E+3nMAssay Description:Binding activity against dopamine receptor D2 in rat brain, using [3H]spiperone as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed