BDBM50023316 2-Isopropyl-8-[(4-pyridin-3-yl-butylamino)-methyl]-pyrido[2,1-b]quinazolin-11-one::CHEMBL141818

SMILES CC(C)c1ccc2nc3ccc(CNCCCCc4cccnc4)cn3c(=O)c2c1

InChI Key InChIKey=RGNIRBZAYFBIKC-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50023316   

TargetPlatelet-activating factor receptor(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50023316(2-Isopropyl-8-[(4-pyridin-3-yl-butylamino)-methyl]...)
Affinity DataIC50: 1.00E+3nMAssay Description:Ability to inhibit platelet activating factor (PAF) binding to platelets by 50% was determined by using [3H]PAF as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed