BDBM50024211 (+/-)2-(3-Methoxy-phenyl)-1-methyl-ethylamine::2-(3-Methoxy-phenyl)-1-methyl-ethylamine::2-(3-Methoxy-phenyl)-1-methyl-ethylamine(MMA)::CHEMBL16247

SMILES COc1cccc(CC(C)N)c1

InChI Key InChIKey=VEJWNIYARKAHFI-UHFFFAOYSA-N

Data  7 KI  1 Kd

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 8 hits for monomerid = 50024211   

Target5-hydroxytryptamine receptor 2B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50024211(2-(3-Methoxy-phenyl)-1-methyl-ethylamine(MMA) | (+...)
Affinity DataKd:  1.20E+3nMAssay Description:Affinity against 5-hydroxytryptamine 2B receptor in the isolated rat stomach fundusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
LigandPNGBDBM50024211(2-(3-Methoxy-phenyl)-1-methyl-ethylamine(MMA) | (+...)
Affinity DataKi:  2.66E+3nMAssay Description:Evaluated for binding affinity towards rat cortical membranes at 5-hydroxytryptamine 1 receptor binding site by using [3H]-5-HT as a radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
LigandPNGBDBM50024211(2-(3-Methoxy-phenyl)-1-methyl-ethylamine(MMA) | (+...)
Affinity DataKi:  2.66E+3nMAssay Description:Binding affinity for 5-hydroxytryptamine 1 receptor of rat prefrontal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2018
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50024211(2-(3-Methoxy-phenyl)-1-methyl-ethylamine(MMA) | (+...)
Affinity DataKi:  7.85E+3nMAssay Description:Binding affinity to rat cortical membranes at 5-hydroxytryptamine 2 (5-HT2) receptor using [3H]KET as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50024211(2-(3-Methoxy-phenyl)-1-methyl-ethylamine(MMA) | (+...)
Affinity DataKi:  7.85E+3nMAssay Description:Displacement of [3H]ketanserin from rat prefrontal cortex 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50024211(2-(3-Methoxy-phenyl)-1-methyl-ethylamine(MMA) | (+...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]mesulergine from A9 cells stably expressing rat 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50024211(2-(3-Methoxy-phenyl)-1-methyl-ethylamine(MMA) | (+...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]ketanserin from NIH3T3 cells stably expressing rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50024211(2-(3-Methoxy-phenyl)-1-methyl-ethylamine(MMA) | (+...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A expressed in mouse NIH/3T3 cell membranes after 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2019
Entry Details Article
PubMed