BDBM50035926 CHEMBL3361079

SMILES Cc1cccc2c(cc(C(=O)c3ccc(Cl)cc3)n12)C(=O)NCC#C

InChI Key InChIKey=RPLQRYPCSHTXPG-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50035926   

TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Human)
Alexandru Ioan Cuza University

Curated by ChEMBL

LigandBDBM50035926(CHEMBL3361079)Copy SMILESCopy InChI

Affinity DataIC50: 1.49E+4nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
3/15/2016
Entry Details Article
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