BDBM50036274 CHEMBL3361086

SMILES Cc1cccc2c(cc(C(=O)c3ccc(Br)cc3)n12)C(=O)OCC#C

InChI Key InChIKey=GHIYZOAWPOFIFT-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50036274   

TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Human)
Alexandru Ioan Cuza University

Curated by ChEMBL

LigandBDBM50036274(CHEMBL3361086)Copy SMILESCopy InChI

Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human recombinant farnesyltransferase using octyl-beta-D-glucopyranoside as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
3/15/2016
Entry Details Article
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