BDBM50036530 CHEMBL3353589

SMILES OC(=O)c1ccc(cc1)S(=O)(=O)N(CCCc1ccccc1)c1ncc(cc1Cl)C(F)(F)F

InChI Key InChIKey=ONCWBUXXMWVYOW-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50036530   

TargetTransient receptor potential cation channel subfamily M member 8(Human)
Raqualia Pharma

Curated by ChEMBL

LigandBDBM50036530(CHEMBL3353589)Copy SMILESCopy InChI

Affinity DataIC50: 49nMAssay Description:Antagonist activity at human TRPM8 expressed in HEK293 cells assessed as inhibition of menthol induced Ca2+ influxMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPurchaseCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
3/15/2016
Entry Details Article
Copy Entry DOIPubMed
Copy Rxn URL