BDBM50036559 CHEMBL3353584

SMILES Cc1cc(cnc1N(Cc1ccccc1)S(=O)(=O)c1ccc(cc1)C(O)=O)C(F)(F)F

InChI Key InChIKey=QSHZUPQNJLCBOA-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50036559   

TargetTransient receptor potential cation channel subfamily M member 8(Human)
Raqualia Pharma

Curated by ChEMBL

LigandBDBM50036559(CHEMBL3353584)Copy SMILESCopy InChI

Affinity DataIC50: 736nMAssay Description:Antagonist activity at human TRPM8 expressed in HEK293 cells assessed as inhibition of menthol induced Ca2+ influxMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
3/15/2016
Entry Details Article
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