BDBM50058783 CHEMBL3335135

SMILES FC(F)(F)c1ccc(NC(=O)c2ccc(CN3CCOCC3)cc2)cc1

InChI Key InChIKey=FGDAZKGJPZGOKI-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50058783   

TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Human)
Eisai

Curated by ChEMBL

LigandBDBM50058783(CHEMBL3335135)Copy SMILESCopy InChI

Affinity DataIC50: 280nMAssay Description:Inhibition of HIF1 signaling in human U251 cells expressing VEGF by VEGF promoter-driven PLAP reporter gene assayMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPurchaseCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
4/2/2016
Entry Details Article
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