BDBM50059586 CHEMBL406338::N-allyl[D-Pro-10]Dyn A-(1-11)
SMILES CC[C@H](C)[C@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@H](Cc1ccc(O)cc1)NCC=C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCCCN)C(O)=O
InChI Key InChIKey=MKKPRLAUMQVIGT-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50059586
Affinity DataIC50: 2.30nMAssay Description:Binding affinity towards Opioid receptor kappa 1 using [3H]diprenorphine as radioligand in guinea pig cerebellar membrane in absence of 120 mM NaCl +...More data for this Ligand-Target Pair
Affinity DataIC50: 229nMAssay Description:Binding affinity towards Opioid receptor kappa 1 using [3H]diprenorphine as radioligand in guinea pig cerebellar membrane in presence of 120 mM NaCl ...More data for this Ligand-Target Pair
Affinity DataKi: 0.0490nMAssay Description:Affinity against Opioid receptor kappa 1 was determined by measuring the inhibition of [3H]bremazocine binding to guinea pig cerebellar membranesMore data for this Ligand-Target Pair
Affinity DataKi: 10.9nMAssay Description:Affinity against Opioid receptor mu 1 was determined by measuring the inhibition of [3H]DAMGO binding to rat forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 499nMAssay Description:Affinity against Opioid receptor delta 1 was determined by measuring the inhibition of [3H]DPDPE binding to rat forebrain membranesMore data for this Ligand-Target Pair