BDBM50064356 CHEMBL3403708

SMILES CCCc1c(OCCCCN2C(=O)N(C)C(C)(C)C2=O)ccc2c(cc(=O)oc12)C(F)(F)F

InChI Key InChIKey=AIPZKNVPWAZNKM-UHFFFAOYSA-N

Data  4 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50064356   

TargetOxysterols receptor LXR-beta(Human)
Kowa

Curated by ChEMBL
LigandPNGBDBM50064356(CHEMBL3403708)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at LXRbeta (unknown origin) expressed in CHOK1 cells incubated for 24 hrs by GAL4-responsive luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Human)
Kowa

Curated by ChEMBL
LigandPNGBDBM50064356(CHEMBL3403708)
Affinity DataEC50:  1.02E+3nMAssay Description:Agonist activity at Gal4-tagged LXRbeta (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Kowa

Curated by ChEMBL
LigandPNGBDBM50064356(CHEMBL3403708)
Affinity DataEC50:  2.40E+3nMAssay Description:Agonist activity at LXRalpha (unknown origin) expressed in CHOK1 cells incubated for 24 hrs by GAL4-responsive luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Kowa

Curated by ChEMBL
LigandPNGBDBM50064356(CHEMBL3403708)
Affinity DataEC50:  2.40E+3nMAssay Description:Agonist activity at Gal4-tagged LXRalpha (unknown origin) expressed in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2016
Entry Details Article
PubMed