BDBM50071857 4-(4-Benzyl-piperazin-1-yl)-1H-indole::CHEMBL328051

SMILES C(N1CCN(CC1)c1cccc2[nH]ccc12)c1ccccc1

InChI Key InChIKey=JLZIBIQTDGMAFZ-UHFFFAOYSA-N

Data  5 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50071857   

TargetD(2) dopamine receptor(Rat)
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071857(4-(4-Benzyl-piperazin-1-yl)-1H-indole | CHEMBL3280...)
Affinity DataKi:  3.20nMAssay Description:Affinity of compound for the Dopamine receptor D2 in rat striatal membranes was determined for low agonist state in rat striatal membranes using [3H]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071857(4-(4-Benzyl-piperazin-1-yl)-1H-indole | CHEMBL3280...)
Affinity DataKi:  15nMAssay Description:Affinity towards human Dopamine receptor D4.4 expressed in CHO cells using [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071857(4-(4-Benzyl-piperazin-1-yl)-1H-indole | CHEMBL3280...)
Affinity DataKi:  17nMAssay Description:Affinity of compound for the Dopamine receptor D2 in rat striatal membranes was determined for low antagonist state in rat striatal membranes using [...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071857(4-(4-Benzyl-piperazin-1-yl)-1H-indole | CHEMBL3280...)
Affinity DataKi:  35nMAssay Description:Affinity towards human Dopamine receptor D3 expressed in CHO cells using [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Wyeth-Ayerst Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50071857(4-(4-Benzyl-piperazin-1-yl)-1H-indole | CHEMBL3280...)
Affinity DataKi:  53nMAssay Description:Affinity towards human Dopamine receptor D2 expressed in CHO cells using [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed