BDBM50071991 1-(2,2,4-Trimethyl-2,10-dihydro-1H-indeno[1,2-g]quinolin-8-yl)-ethanone::1-(2,2,4-trimethyl-2,10-dihydro-1H-indeno[1,2-g]quinolin-8-yl)ethanone::CHEMBL93345

SMILES CC(=O)c1ccc-2c(Cc3cc4NC(C)(C)C=C(C)c4cc-23)c1

InChI Key InChIKey=QROLJIOISIOIPO-UHFFFAOYSA-N

Data  2 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50071991   

TargetProgesterone receptor(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071991(1-(2,2,4-trimethyl-2,10-dihydro-1H-indeno[1,2-g]qu...)
Affinity DataIC50: 164nMAssay Description:Antagonist activity against human progesterone receptor B (hPR-B) in co-transfected CV-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071991(1-(2,2,4-trimethyl-2,10-dihydro-1H-indeno[1,2-g]qu...)
Affinity DataKi:  176nMAssay Description:Binding affinity against human progesterone receptor-A (hPR-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071991(1-(2,2,4-trimethyl-2,10-dihydro-1H-indeno[1,2-g]qu...)
Affinity DataKi:  178nMAssay Description:Displacement of [3H]progesterone from Progesterone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed