BDBM50075231 (5-Bromo-2-{3-[2-(4-dimethylamino-piperidin-1-yl)-ethyl]-benzo[b]thiophen-2-ylmethoxy}-phenyl)-methanol::CHEMBL145056

SMILES CN(C)C1CCN(CCc2c(COc3ccc(Br)cc3CO)sc3ccccc23)CC1

InChI Key InChIKey=VSDGMNFJZBSRSC-UHFFFAOYSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50075231   

TargetNeuropeptide Y receptor type 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50075231((5-Bromo-2-{3-[2-(4-dimethylamino-piperidin-1-yl)-...)
Affinity DataKi:  15nMAssay Description:Functional Neuropeptide Y receptor type 1 antagonism was evaluated by its ability to reverse NPY induced inhibition of forskolin-stimulated cyclic AM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50075231((5-Bromo-2-{3-[2-(4-dimethylamino-piperidin-1-yl)-...)
Affinity DataKi:  15nMAssay Description:Ability to displace [125I]pPYY from AV12 cell line stably transfected with cloned human neuropeptide Y receptor type 1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed