BDBM50089267 CHEMBL3577893

SMILES C[C@@H](N(Cc1cc(ccc1F)C(O)=O)C(=O)c1cnc2ccccc2c1)c1ccc(F)cc1

InChI Key InChIKey=BYFNPEHCGXRBNW-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50089267   

TargetTransient receptor potential cation channel subfamily M member 8(Human)
Pfizer

Curated by ChEMBL

LigandBDBM50089267(CHEMBL3577893)Copy SMILESCopy InChI

Affinity DataIC50: 446nMAssay Description:Antagonist activity against human recombinant TRPM8 expressed in CHO T-rex cells assessed as inhibition of WS12-induced calcium response pre-incubate...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
10/8/2016
Entry Details Article
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