BDBM50095345 CHEMBL3589910

SMILES Nc1nc(NC(=O)c2ccccc2)ccc1-c1ccccc1OC(F)(F)F

InChI Key InChIKey=KVHIYIURFFIYHO-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50095345   

TargetSodium channel protein type 10 subunit alpha(Human)
Pfizer

Curated by ChEMBL

LigandBDBM50095345(CHEMBL3589910)Copy SMILESCopy InChI

Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of human Nav1.8 expressed in HEK293 cells assessed as reduction in blue fluorescent signal by VSP-FRET assayMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
10/16/2016
Entry Details Article
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