BDBM50098012 2-(1-Ethyl-2-phenyl-1H-indol-3-yl)-N-isopropyl-N-pyridin-4-ylmethyl-acetamide::CHEMBL352831

SMILES CCn1c(c(CC(=O)N(Cc2ccncc2)C(C)C)c2ccccc12)-c1ccccc1

InChI Key InChIKey=CRMSUCZMVYPRIO-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50098012   

TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Human)
Merck Research Laboratories

Curated by ChEMBL

LigandBDBM50098012(2-(1-Ethyl-2-phenyl-1H-indol-3-yl)-N-isopropyl-N-p...)Copy SMILESCopy InChI

Affinity DataIC50: 3.80E+3nMAssay Description:Concentration required for the inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
10/5/2012
Entry Details Article
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