BDBM50098016 CHEMBL171214::N-Cyclopropyl-2-(2-phenyl-1H-indol-3-yl)-N-pyridin-4-ylmethyl-acetamide

SMILES O=C(Cc1c([nH]c2ccccc12)-c1ccccc1)N(Cc1ccncc1)C1CC1

InChI Key InChIKey=RMWSUCRYTTWVOL-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50098016   

TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Human)
Merck Research Laboratories

Curated by ChEMBL

LigandBDBM50098016(N-Cyclopropyl-2-(2-phenyl-1H-indol-3-yl)-N-pyridin...)Copy SMILESCopy InChI

Affinity DataIC50: 171nMAssay Description:Concentration required for the inhibitory activity against human FarnesyltransferaseMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
10/5/2012
Entry Details Article
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