BDBM50099263 3-(1-Methyl-piperidin-2-yl)-2-phenyl-1H-indole::3-(1-Methylpiperidin-2-yl)-2-phenyl-1H-indole::CHEMBL43697

SMILES CN1CCCCC1c1c([nH]c2ccccc12)-c1ccccc1

InChI Key InChIKey=YKKPUIDGSXNPRO-UHFFFAOYSA-N

Data  5 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50099263   

Target5-hydroxytryptamine receptor 2A(Human)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099263(3-(1-Methylpiperidin-2-yl)-2-phenyl-1H-indole | 3-...)
Affinity DataKi:  14nMAssay Description:Ability to displace [3H]ketanserin binding to human 5-hydroxytryptamine 2A receptor stably expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099263(3-(1-Methylpiperidin-2-yl)-2-phenyl-1H-indole | 3-...)
Affinity DataKi: >1.70E+3nMAssay Description:Ability to displace [3H]spiperone binding to CHO cells stably expressing dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099263(3-(1-Methylpiperidin-2-yl)-2-phenyl-1H-indole | 3-...)
Affinity DataKi:  2.00E+3nMAssay Description:Ability to displace [3H]mesulergine binding to human 5-hydroxytryptamine 2C receptor stably expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50099263(3-(1-Methylpiperidin-2-yl)-2-phenyl-1H-indole | 3-...)
Affinity DataKi:  7.00E+3nMAssay Description:Inhibition of human ERG channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
LigandPNGBDBM50099263(3-(1-Methylpiperidin-2-yl)-2-phenyl-1H-indole | 3-...)
Affinity DataKi:  7.00E+3nMAssay Description:Displacement of [3H]dofetilide from HEK cells expressing hERG voltage dependent IKr potassium channel Kv11.1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed