BDBM50108390 4-Amino-5-chloro-2-methoxy-N-(2-methyl-2-aza-bicyclo[2.2.2]oct-5-yl)-benzamide::CHEMBL56994

SMILES COc1cc(N)c(Cl)cc1C(=O)NC1CC2CCC1CN2C

InChI Key InChIKey=KAVKRBZLNSOOJY-UHFFFAOYSA-N

Data  2 KI  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50108390   

Target5-hydroxytryptamine receptor 4(Guinea pig)
Universidad De Alcal£

Curated by ChEMBL
LigandPNGBDBM50108390(4-Amino-5-chloro-2-methoxy-N-(2-methyl-2-aza-bicyc...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity towards 5-HT4 receptor in striatum membranes of guinea-pig brain was evaluatedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Universidad De Alcal£

Curated by ChEMBL
LigandPNGBDBM50108390(4-Amino-5-chloro-2-methoxy-N-(2-methyl-2-aza-bicyc...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity towards 5-HT3 receptor in rat was evaluatedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Universidad De Alcal£

Curated by ChEMBL
LigandPNGBDBM50108390(4-Amino-5-chloro-2-methoxy-N-(2-methyl-2-aza-bicyc...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity towards 5-HT3 receptor in rat was evaluatedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Universidad De Alcal£

Curated by ChEMBL
LigandPNGBDBM50108390(4-Amino-5-chloro-2-methoxy-N-(2-methyl-2-aza-bicyc...)
Affinity DataKi:  130nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat was evaluatedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Universidad De Alcal£

Curated by ChEMBL
LigandPNGBDBM50108390(4-Amino-5-chloro-2-methoxy-N-(2-methyl-2-aza-bicyc...)
Affinity DataKi:  842nMAssay Description:Binding affinity towards D2 receptor in rat was evaluatedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2012
Entry Details Article
PubMed