BDBM50111899 5-(2-Ethoxy-phenyl)-1-methyl-3-propyl-1,6-dihydro-pyrazolo[4,3-d]pyrimidin-7-one::5-(2-ethoxyphenyl)-1-methyl-3-propyl-1H-pyrazolo[4,3-d]pyrimidin-7(6H)-one::CHEMBL54079

SMILES CCCc1nn(C)c2c1nc([nH]c2=O)-c1ccccc1OCC

InChI Key InChIKey=MXQUEDUMKWBYHI-UHFFFAOYSA-N

Data  11 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 11 hits for monomerid = 50111899   

LigandPNGBDBM50111899(5-(2-ethoxyphenyl)-1-methyl-3-propyl-1H-pyrazolo[4...)
Affinity DataIC50: 27nMAssay Description:Inhibition of Phosphodiesterase 5 from human corpus cavernosumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50111899(5-(2-ethoxyphenyl)-1-methyl-3-propyl-1H-pyrazolo[4...)
Affinity DataIC50: 40nMAssay Description:Inhibition of Phosphodiesterase 5More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50111899(5-(2-ethoxyphenyl)-1-methyl-3-propyl-1H-pyrazolo[4...)
Affinity DataIC50: 500nMAssay Description:Inhibition of Phosphodiesterase 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50111899(5-(2-ethoxyphenyl)-1-methyl-3-propyl-1H-pyrazolo[4...)
Affinity DataIC50: 500nMAssay Description:Inhibition of Phosphodiesterase 3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50111899(5-(2-ethoxyphenyl)-1-methyl-3-propyl-1H-pyrazolo[4...)
Affinity DataIC50: 790nMAssay Description:Inhibition of phosphodiesterase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50111899(5-(2-ethoxyphenyl)-1-methyl-3-propyl-1H-pyrazolo[4...)
Affinity DataIC50: 27nMAssay Description:Inhibition of phosphodiesterase 5More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50111899(5-(2-ethoxyphenyl)-1-methyl-3-propyl-1H-pyrazolo[4...)
Affinity DataIC50: 39.8nMAssay Description:Inhibition of PDE5More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandPNGBDBM50111899(5-(2-ethoxyphenyl)-1-methyl-3-propyl-1H-pyrazolo[4...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Phosphodiesterase 3 from rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50111899(5-(2-ethoxyphenyl)-1-methyl-3-propyl-1H-pyrazolo[4...)
Affinity DataIC50: 790nMAssay Description:Inhibition of Phosphodiesterase 1 from rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50111899(5-(2-ethoxyphenyl)-1-methyl-3-propyl-1H-pyrazolo[4...)
Affinity DataIC50: 27nMAssay Description:Inhibition of Phosphodiesterase 5 from rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50111899(5-(2-ethoxyphenyl)-1-methyl-3-propyl-1H-pyrazolo[4...)
Affinity DataIC50: 27nMAssay Description:Inhibition of human corpus cavernosum PDE5More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed