BDBM50126167 CHEMBL3629675

SMILES FC(F)(F)c1ccc2CCNC(=O)c2c1

InChI Key InChIKey=PWZSJDNHPNHZMD-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50126167   

TargetProtein mono-ADP-ribosyltransferase PARP10(Human)
Oregon Health & Science University

Curated by ChEMBL
LigandPNGBDBM50126167(CHEMBL3629675)
Affinity DataIC50: 6.55E+4nMAssay Description:Inhibition of PARP-10 L926G mutant (unknown origin) mediated ADP-ribosylation of SRPK2 by fluorescence analysis using 3 uM SRPK2 as a substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2016
Entry Details Article
PubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Human)
Oregon Health & Science University

Curated by ChEMBL
LigandPNGBDBM50126167(CHEMBL3629675)
Affinity DataIC50: 6.61E+4nMAssay Description:Inhibition of PARP-10 L926G mutant (unknown origin) mediated ADP-ribosylation of SRPK2 by fluorescence analysis using 3 uM SRPK2 as a substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2016
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Oregon Health & Science University

Curated by ChEMBL
LigandPNGBDBM50126167(CHEMBL3629675)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PARP1 (unknown origin) by fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2016
Entry Details Article
PubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Human)
Oregon Health & Science University

Curated by ChEMBL
LigandPNGBDBM50126167(CHEMBL3629675)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PARP-10 (unknown origin) mediated ADP-ribosylation of SRPK2 by fluorescence analysis using 3 uM SRPK2 as a substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2016
Entry Details Article
PubMed