BDBM50126558 4-[5-({4-[4-(5-Chloro-thiophene-2-carbonyl)-piperazin-1-yl]-phenylamino}-methyl)-imidazol-1-ylmethyl]-benzonitrile::CHEMBL36192

SMILES Clc1ccc(s1)C(=O)N1CCN(CC1)c1ccc(NCc2cncn2Cc2ccc(cc2)C#N)cc1

InChI Key InChIKey=ZFDLOBWFRTYYFH-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50126558   

TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bovine)
Centre De Recherche Pierre Fabre

Curated by ChEMBL

LigandBDBM50126558(4-[5-({4-[4-(5-Chloro-thiophene-2-carbonyl)-pipera...)Copy SMILESCopy InChI

Affinity DataIC50: 70nMAssay Description:Inhibit of purified bovine Farnesyl protein transferase.More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
10/9/2012
Entry Details Article
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