BDBM50132895 CHEMBL115999::Cyclopropylmethyl-[3-(2,4-dichloro-phenyl)-2-ethyl-5-methyl-2H-pyrazolo[4,3-b]pyridin-7-yl]-propyl-amine

SMILES CCCN(CC1CC1)c1cc(C)nc2c(-c3ccc(Cl)cc3Cl)n(CC)nc12

InChI Key InChIKey=KFDFFNFTGSLBLC-UHFFFAOYSA-N

Data  1 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50132895   

TargetCorticotropin-releasing factor receptor 1(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50132895(Cyclopropylmethyl-[3-(2,4-dichloro-phenyl)-2-ethyl...)
Affinity DataKi:  46nMAssay Description:Compound was tested to inhibit Corticotropin releasing factor receptor 1-stimulated c-AMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed