BDBM50139471 CHEMBL3763770

SMILES Clc1ccc(cc1)-c1csc(NCc2cn(Cc3ccc(cc3)C#N)cn2)c1C#N

InChI Key InChIKey=GTWJDPOBPWEGMS-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50139471   

TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Human)
Cnrs Upr2301

Curated by ChEMBL

LigandBDBM50139471(CHEMBL3763770)Copy SMILESCopy InChI

Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesyl pyrophosphate and Dansyl-GCVLS peptide after 15 mins by fluorescence assayMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
6/2/2017
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