BDBM50144146 ({3-methoxy-9-phenyl-8-oxatricyclo[8.4.0.0^{2,7}]tetradeca-1(10),2,4,6,11,13-hexaen-12-yl}sulfamoyl)dimethylamine::CHEMBL62118

SMILES COc1cccc2OC(c3ccccc3)c3cc(NS(=O)(=O)N(C)C)ccc3-c12

InChI Key InChIKey=SDBUTPFXNGKELI-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50144146   

TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144146(({3-methoxy-9-phenyl-8-oxatricyclo[8.4.0.0^{2,7}]t...)
Affinity DataIC50: 41nMAssay Description:Displacement of [3H]dexamethasone from human Glucocorticoid receptor (GR); Value ranges from 26-67 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144146(({3-methoxy-9-phenyl-8-oxatricyclo[8.4.0.0^{2,7}]t...)
Affinity DataIC50: 121nMAssay Description:Displacement of [3H]dexamethasone from human Glucocorticoid receptor (GR); Value ranges from 150-220 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed