BDBM50149210 CHEMBL3769994

SMILES Nc1ccc2c(nc(nc2c1)-c1cnc(N)nc1)N1CCOCC1

InChI Key InChIKey=HOAHRWMUDCKNPY-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50149210   

TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Sun Yat-Sen University

Curated by ChEMBL

LigandBDBM50149210(CHEMBL3769994)Copy SMILESCopy InChI

Affinity DataIC50: 49nMAssay Description:Inhibition of PI3K alpha (unknown origin) using PIP2 as substrate after 1 hr by kinase-Glo luminescent assayMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
6/23/2017
Entry Details Article
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