BDBM50149906 CHEMBL3770104

SMILES Cc1cc(C)c(CNC(=O)c2ccc3cnn(C4CCCC4)c3c2C)c(=O)[nH]1

InChI Key InChIKey=WEIMXAIORJYAGU-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50149906   

TargetHistone-lysine N-methyltransferase EZH2(Human)
Epizyme

Curated by ChEMBL
LigandPNGBDBM50149906(CHEMBL3770104)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of methyltransferase activity of human EZH2 using chicken oligonucleotide as substrate by pull down assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2017
Entry Details Article
PubMed