BDBM50154520 CHEMBL3775050

SMILES Fc1ccc(-c2c[nH]c(n2)[C@H]2Cc3c([nH]c4ccccc34)[C@H](N2)C2CCOCC2)c(F)c1

InChI Key InChIKey=GAGIZVXQARBUAM-UHFFFAOYSA-N

Data  2 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50154520   

TargetSomatostatin receptor type 3(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50154520(CHEMBL3775050)
Affinity DataIC50: 23nMAssay Description:Binding affinity to human somatostatin receptor type 3More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2017
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50154520(CHEMBL3775050)
Affinity DataEC50:  37nMAssay Description:Antagonist activity at human somatostatin receptor type 3 assessed as inhibition of cAMP levelsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2017
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50154520(CHEMBL3775050)
Affinity DataIC50: 634nMAssay Description:Binding affinity to human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2017
Entry Details Article
PubMed