BDBM50155455 3-(4-Iodo-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid (2-fluoro-ethyl)-amide::CHEMBL183259

SMILES CN1C2CCC1C(C(C2)c1ccc(I)cc1)C(=O)NCCF

InChI Key

Data  3 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50155455   

TargetSodium-dependent serotonin transporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155455(3-(4-Iodo-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oct...)
Affinity DataKi:  30.8nMAssay Description:Displacement of [3H]cyanoimiprimine from serotonin transporter of rat cerebral cortical homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155455(3-(4-Iodo-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oct...)
Affinity DataKi:  44.5nMAssay Description:Displacement of [3H]CIT from dopamine transporter of rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50155455(3-(4-Iodo-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oct...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-nisoxetine from norepinephrine transporter of rat cerebral corticex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed